aripiprazole lauroxil
Ligand Summary
prodrug of aripiprazole, following intramuscular injection is converted by enzyme-mediated hydrolysis to N-hydroxymethyl aripiprazole which is then hydrolyzed to aripiprazole
UNII: B786J7A343
PubChem: 49831411
ChEMBL: CHEMBL2219425
DrugCentral: 5052
LyCHI: 3FT39PUS83SK
Target Activities
4 Activities
Items per page:
10
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | PARTIAL AGONIST | |||||
Ki | PARTIAL AGONIST | |||||
Ki | ANTAGONIST | |||||
Ki | ||||||